平安! 发表于 2011-11-9 19:57 8 K, N: V8 o; F$ d+ c5 Z7 n
Pazopanib (100 mg/kg/day free base equivalent) 1 j" r6 b T, w* P/ c% V
这是个已经在美国上市的老药了,能下载到正式药物使用说明书英文版。" |+ z' P% H0 V( b" N
搜索了一下,原料一大堆。
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4 n3 b- r& G* R/ k2 j对不起!100mg/kg是用于移植瘤的,我弄错了。
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以下是正版说明书的推荐用量。/ J% r6 N8 f N
7 f7 _3 s. J; g/ M3 T--------------------- DOSAGE AND ADMINISTRATION ----------------
5 k# E5 |# D% ?& X9 s* 800 mg orally once daily without food (at least 1 hour before or 2 hours after a meal). (2.1) 2 k7 W b* T9 V
* Baseline moderate hepatic impairment – 200 mg orally once daily. Not recommended in patients with severe hepatic impairment. (2.2) 0 q* ?( R8 @' [
---------------------DOSAGE FORMS AND STRENGTHS --------------& y$ ?; A6 [! L: C$ d
200 mg tablets. (3)
" Z N0 Q: _/ P4 a/ c" B) h) A/ {6 c! m-------------------------------CONTRAINDICATIONS------------------------ |